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產品編號:4083600
純度規格:
包裝規格:10 MG
產品編號:4083599
純度規格:A cell permeable, brain permeant antagonist of polypeptide chemokine prokineticin 2 receptor (IC50 = 5 nM and 8.2 nM for PKR1 and PKR2, respectively).
包裝規格:5 MG
產品編號:4083597
純度規格:
包裝規格:2 MG
產品編號:4083596
純度規格:A cell permeable competitive inhibitor of Pin1 (EC50 = 4.1 μM, Ki = 50 nM).
包裝規格:10 MG
產品編號:4083594
純度規格:A cell-permeable, potent and competitive inhibitor of fructose-2,6-bisphosphatase 3 (PFKFB3; IC50 = 670 nM).
CAS NO:75187-63-2
包裝規格:25 MG
產品編號:4083593
純度規格:A cell-permeable inhibitor of PFKFB3 that reversibly docks to its substrate binding domain (IC50 = 207 nM)
包裝規格:25 MG
產品編號:4083592
純度規格:A cell-permeable nematicidal compound that covalently binds to the peroxidatic cysteine of peroxiredoxin II in T. gondii and irreversibly blocks its hyperperoxidation activity (IC50 = 23 μM).
CAS NO:18080-67-6
包裝規格:25 MG
產品編號:4083589
純度規格:A cell-permeable, selective &direct blocker of p18-Cdk6 interaction. Inhibits p18INK4C protein activity &favors HSCs self-renewal by ~4.2-fold.
CAS NO:77408-67-4
包裝規格:25 MG
產品編號:4083588
純度規格:A cell-permeable compound with cytotoxicity towards quiescent cells in colon cancer 3-D microtissues (~ 6 μM). Reduces mitochondrial oxidative phosphorylation in tumor cells.
包裝規格:10 MG
產品編號:4083587
純度規格:Prevents melanopsin/Opn4 photoactivation in a reversible manner. Inhibits cellular phototransduction mediated by human Opn4 (IC50 = 665 nM; using CHO transfectants).
CAS NO:457961-34-1
包裝規格:10 MG
產品編號:4083585
純度規格:
包裝規格:10 MG
產品編號:4083584
純度規格:A potent activator of Ca2+ -activated K+ channels of SK and IK types, but not BK type channels. It is at least 1000 times more potent than 1-EBIO.
CAS NO:18711-16-5
包裝規格:10 MG
產品編號:4083583
純度規格:A cell-permeable, potent Nrf-2 activator that stimulates HO-1 expression in murine microglial BV-2 cultures. Induces overall Nrf2 cellular accumulation and nuclear translocation.
包裝規格:10 MG
產品編號:4083582
純度規格:A cell-permeable inhibitor of nonsense-mediated mRNA decay (NMD) that enhances the stability of premature termination codon mutated p53 mRNA in N417 and HDQP-1 cells.
包裝規格:10 MG
產品編號:4083581
純度規格:A cell-potent, bioavailable NLRP3 inflammasome activation inhibitor. Effectively blocks caspase-1 &-11 activation, IL-1β processing and IL-1β &IL-6 secretion.
CAS NO:256373-96-3
包裝規格:10 MG
產品編號:4083578
純度規格:
包裝規格:25 MG
產品編號:4083577
純度規格:A cell-permeable neomycin derived artificial nucleobase conjugate. Inhibits the production of oncogenic miRNAs 372 (IC50 = 2.4 μM) by binding to pre-miRNAs and interrupts processing by Dicer.
包裝規格:2 MG
產品編號:4083576
純度規格:A blood-brain barrier permeable, potent, selective, and reversible antagonist of mGlu7 receptor (IC50 = 3.5 and 2.8 μM for mGlu7a and mGlu7b in CHO cells).
CAS NO:196928-50-4
包裝規格:10 MG
產品編號:4083575
純度規格:A cell-permeable, bioavailable, highly potent inhibitor of acyl CoA:monoacylglycerol acyltransferase 2 inhibitor (MGAT2, IC50 = 3.4 nM). Displays good microsomal stability.
包裝規格:5 MG
產品編號:4083573
純度規格:
包裝規格:10 MG
產品編號:4083571
純度規格:A synthetic cyclic alkylaminoluciferin with properties superior to D-luciferin. Binds to luciferase with higher affinity.
包裝規格:10 MG
產品編號:4083570
純度規格:A cell-permeable stain for neutral lipids. Does not stain phospholipids.
包裝規格:5 MG
產品編號:4083569
純度規格:
包裝規格:5 MG
產品編號:4083567
純度規格:A cell-permeable compound that prevents various bacterial toxins from exerting their cytotoxic activity by blocking endosomal trafficking/maturation into acidified late endosomes.
包裝規格:25 MG
產品編號:4083565
純度規格:A fast acting, reversible, and selective activator of Kir6.2/SUR1 channels (EC50 = 7 μM).
包裝規格:10 MG
產品編號:4083563
純度規格:A cell-permeable, direct, non-covalent inhibitor of Keap1-Nrf2 protein-protein interaction (Kd = 1 μM) that causes the dissociation of Nrf2 from keap1 in the cytosol.
包裝規格:10 MG
產品編號:4083562
純度規格:
包裝規格:10 MG
產品編號:4083561
純度規格:
包裝規格:5 MG
產品編號:4083560
純度規格:A cell-permeable, superior inhibitor of Jumonji C domain histone lysine demethylase. About 30 fold more potent than IOX1 (EC50 = 3.8 μM for KDM4A in HeLa cells vs. 100 μM for IOX1).
包裝規格:10 MG
產品編號:4083558
純度規格:A cell permeable analog of curcumin that acts as a specific inhibitor of JAK2 (~ 5 μM) and blocks STAT3 phosphorylation in MDA-MB-231 and PANC-1 cancer cells.
包裝規格:25 MG
產品編號:4083557
純度規格:The cell-permeable, selective inhibitor of eIF2α/eIF2S1 Ser51 phosphorylation-initiated UPR response (~25 to 200 nM) upon ER stress induction.
包裝規格:10 MG
產品編號:4083556
純度規格:InSolutionTM Y-27632, Sterile-Filtered, Cell Culture-Tested, CAS 146986-50-7, is a 10 mM sterile-filtered solution of Y-27632 in H2O. Acts as an inhibitor of Rho kinases (Ki = 140 nM for p160ROCK).
CAS NO:146986-50-7
包裝規格:2 MG
產品編號:4083555
純度規格:A 25 mM (2 mg/221 μL) sterile-filtered solution of TLR4 Inhibitor, TAK-242 in DMSO.
CAS NO:243984-11-4
包裝規格:2 MG
產品編號:4083553
純度規格:A 25 mM (10 mg/650 μl) sterile-filtered solution of SRT1720, HCl in DMSO.
CAS NO:1001645-58-4
包裝規格:10 MG
產品編號:4083552
純度規格:A 25 μM (10 mg/583 μL) sterile-filtered solution of Pepstatin A, Synthetic in DMSO.
CAS NO:26305-03-3
包裝規格:10 MG
產品編號:4083551
純度規格:
CAS NO:1135280-28-2
包裝規格:500 μG
產品編號:4083550
純度規格:
包裝規格:5 MG
產品編號:4083549
純度規格:A 25 mM (1 mg/98 μL) sterile-filtered solution of Histone Methyltransferase EZH2 Inhibitor, DZNep in H2O.
CAS NO:102052-95-9
包裝規格:1 MG
產品編號:4083547
純度規格:A 50 mM (2 mg/106.23 μL) sterile-filtered solution of APT1 Inhibitor, palmostatin B in DMSO.
包裝規格:2 MG
產品編號:4083546
純度規格:A 30 mM (1 mg/98 μL) sterile-filtered solution of Aphidicolin in DMSO.
CAS NO:38966-21-1
包裝規格:1 MG
產品編號:4083545
純度規格:A cell-permeable, selective inhibitor of E3 ligase complex SCFβTrCP1-mediated ubiquitination of phosphorylated IκBα (IC50 = 5.2 μM).
包裝規格:10 MG
產品編號:4083542
純度規格:A cell-permeable inhibitor of isocitrate dehydrogenase 2 R140Q mutant-containing dimers. Has minimal effect on wild type dimer-catalyzed alpha-KG production.
CAS NO:1432660-47-3
包裝規格:10 MG
產品編號:4083539
純度規格:A cell-permeable 6-amino-purine based compound that selectively binds to HSP90a (EC50 = 5.4 μM) and inhibits its activity cancer cells.
包裝規格:5 MG
產品編號:4083534
純度規格:A cell-permeable, highly potent, and selective agonist of free fatty acid receptor 1 (FFA1; GPR40; EC50 = 20 nM in FFA1-transfected HEK-293 cells).
包裝規格:10 MG
產品編號:4083533
純度規格:
包裝規格:10 MG
產品編號:4083532
純度規格:
CAS NO:491833-30-8
包裝規格:10 MG
產品編號:4083527
純度規格:
包裝規格:10 MG
產品編號:4083525
純度規格:A helical 27-mer peptide with E54Q modification that directly binds to EDD (Kd = 320 nM) and disrupts protein-protein interaction of EED with EZH2 and EZH1.
包裝規格:2 MG
產品編號:4083524
純度規格:A cell-permeable inhibitor of Eya2 ED tyrosine phosphatase (IC50 = 4.1 μM; KD = 2.0 μM for hEya2, catalytic domain)
包裝規格:25 MG
產品編號:4083523
純度規格:A cell-permeable compound that reversibly blocks cellular glycosylation and surface expression of Notch, APP, Klotho by blocking events prior to cargo assembly at the ER exit sites.
包裝規格:10 MG
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