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產品編號:4083706
純度規格:A cell-permeable myristoylated hexapeptide that selectively inhibits integrin outside-in signaling without affecting inside-out signaling. Blocks the interaction of Gα3 and integrin β3 subunit.
包裝規格:10 MG
產品編號:4083701
純度規格:A cell-permeable. Reversible, selective inhibitor of the growth of malignant peripheral nerve sheath tumors (EC50 = 439 nM, 754 nM, and 1.0 μM in S462, SNF96.2, and sMPNST cells).
包裝規格:25 MG
產品編號:4083697
純度規格:
包裝規格:10 MG
產品編號:4083692
純度規格:A cell-permeable, potent, selective, reversible inhibitor of Lysine-Specific Demethylase 1 (LSD1; IC50 = 13 nM; Ki = 31 nM).
CAS NO:1423715-09-6
包裝規格:10 MG
產品編號:4083691
純度規格:A cell-permeable, both NADH and pyruvate-competitive isoform A-selective LDH inhibitor. Exhibits enhanced anticancer activity under hypoxic conditions.
CAS NO:1269802-68-7
包裝規格:10 MG
產品編號:4083690
純度規格:A cell-permeable, fast acting, branched polyamine. Induces growth of actin-enriched lamellipodia within minutes without the need for serum cofactors .
包裝規格:10 MG
產品編號:4083688
純度規格:A voltage gated calcium channel gating inhibitor of the dihydropyridine class.
CAS NO:75695-93-1
包裝規格:10 MG
產品編號:4083686
純度規格:A substrate competitive inhibitor of insulin-regulated aminopeptidase (IRAP) activity (Ki = 0.48 μM against 25 μM Leu-AMC).
包裝規格:10 MG
產品編號:4083685
純度規格:A 10 mM (5 mg/1.07 ml) sterile-filtered solution of Wnt Antagonist II, IWP-2) in DMSO.
CAS NO:686770-61-6
包裝規格:5 MG
產品編號:4083683
純度規格:A 25 mM (5 mg/357 μl) sterile-filtered solution of PPACK, 2HCl in H2O.
CAS NO:74392-58-8
包裝規格:5 MG
產品編號:4083680
純度規格:
CAS NO:478336-92-4
包裝規格:10 MG
產品編號:4083678
純度規格:A 50 mM sterile-filtered solution of I-BET in DMSO.
CAS NO:1260907-17-2
包裝規格:5 MG
產品編號:4083677
純度規格:A 25 mM (2 mg/231 μl) sterile-filtered solution of Ginkgolic Acid (15:1) in DMSO.
CAS NO:22910-60-7
包裝規格:2 MG
產品編號:4083676
純度規格:
包裝規格:5 MG
產品編號:4083675
純度規格:
CAS NO:130370-60-4
包裝規格:2 MG
產品編號:4083674
純度規格:A 25 mM solution of (+)-Brefeldin A in DMSO.
CAS NO:20350-15-6
包裝規格:2 MG
產品編號:4083672
純度規格:A cell-permeable compound that competitively binds to Hu antigen R (HuR; Ki = 350 nM) and disrupts the interaction of HuR and adenine- and uridine-rich element (ARE) of target mRNAs.
包裝規格:10 MG
產品編號:4083670
純度規格:
CAS NO:1423058-85-8
包裝規格:10 MG
產品編號:4083667
純度規格:Cell-permeable inhibitor of gp130. Binds to gp130 and induces its phosphorylation at Ser782 in ovarian cancer cells. Suppresses constitutive phosphorylation of and nuclear translocation of Stat3.
包裝規格:10 MG
產品編號:4083664
純度規格:
包裝規格:
產品編號:4083662
純度規格:Specifically binds to the Fn14 surface (Kd = 7.12 mM) and suppresses TWEAK-induced glioma cell migration.
包裝規格:10 MG
產品編號:4083661
純度規格:A cell-permeable structural analog of E1 that acts as an equipotent, SAM-competitive inhibitor of Ezh2/PRC2 inhibitor (Ki = 0.5 to 3 nM against wt &mutant Ezh2-containing PRC2).
包裝規格:5 MG
產品編號:4083658
純度規格:
包裝規格:10 MG
產品編號:4083655
純度規格:DHODH Inhibitor, DSM1, is a highly potent, competitive, tight-binding inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (IC50 = 47 nM; Ki = 15 nM).
包裝規格:25 MG
產品編號:4083653
純度規格:
包裝規格:5 MG
產品編號:4083650
純度規格:
包裝規格:10 MG
產品編號:4083649
純度規格:
CAS NO:1253186-56-9
包裝規格:10 MG
產品編號:4083648
純度規格:A 25 mM (10 mg/608 μL) sterile-filtered solution of CMP-Sialic Acid, Disodium Salt in H2O.
CAS NO:3063-71-6
包裝規格:10 MG
產品編號:4083647
純度規格:
包裝規格:25 MG
產品編號:4083645
純度規格:A cell-permeable, highly potent, and specific inhibitor of CDC-like kinase (CLK; IC50 = 1.1 and 2.4 nM for CLK1 and CLK2, respectively).
包裝規格:5 MG
產品編號:4083644
純度規格:A cell-permeable, potent, irreversible, non-substrate competitive inhibitor of CD45/PTPRC tyrosine phosphatase activity (IC50 = 290 nM).
包裝規格:10 MG
產品編號:4083642
純度規格:Enhances BMP-2 associated signaling by inhibiting Smurf1-mediated Smad1/5 ubiquitination and thereby prolonging the half-life of Smad1 and 5. in 48 h).
包裝規格:10 MG
產品編號:4083641
純度規格:A cell-permeable compound that downregulates cellular BMI-1 levels by inhibiting BMI-1 transcription.
CAS NO:315704-66-6
包裝規格:10 MG
產品編號:4083640
純度規格:A cell permeable, highly potent, selective inhibitor of Aurora A (IC50 = 48 nM). Disrupts MYCN-Aurora A complex.
包裝規格:10 MG
產品編號:4083638
純度規格:A cell-permeable compound that directly and reversibly interacts with miRNA binding domain of Argonaute-2 (Kd = 126 μM) and inhibits binding of miR-20a, miR-26a, miR-107, miR-223 &let-7a to Ago2.
包裝規格:25 MG
產品編號:4083634
純度規格:Acid Ceramidase Inhibitor, BOC, CAS 1644158-57-5, is a cell-permeable, potent inhibitor of acid ceramidase (IC50 = 79 nM against HEK293 lysosomal lysate AC activity).
包裝規格:10 MG
產品編號:4083632
純度規格:An anti-bacterial compound that targets NAD(P)H-dependent enoyl acyl carrier protein reductase (ENR) resulting in the inhibition of bacterial fatty acid synthase.
包裝規格:10 MG
產品編號:4083627
純度規格:A cell-permeable, selective, potent, and reversible inhibitor of USP1-UAF1 deubiquitinase (IC50 = 76 nM in Ub-Rhodamine based assays). Does not disrupt USP1-UAF1 association.
包裝規格:10 MG
產品編號:4083625
純度規格:Directly and selectively binds to the troponin complex in fast skeletal muscle (Kd = 40 nM) and sensitizes it to calcium.
CAS NO:1005491-05-3
包裝規格:10 MG
產品編號:4083624
純度規格:
CAS NO:219766-25-3
包裝規格:25 MG
產品編號:4083622
純度規格:A potent agonist of Toll-like receptor 8 agonist (TLR8, EC50 = 200 nM).
包裝規格:10 MG
產品編號:4083621
純度規格:
包裝規格:10 MG
產品編號:4083618
純度規格:A cell-permeable compound that prevents the transfer of SUMO from the E2 thioester to the substrate without affecting SUMO-activating enzyme E1 (SAE-1/2) or E2 Ubc9-SUMO thioester formation.
包裝規格:10 MG
產品編號:4083617
純度規格:
CAS NO:179386-44-8
包裝規格:5 MG
產品編號:4083616
純度規格:
CAS NO:209986-17-4
包裝規格:250 μG
產品編號:4083615
純度規格:A cell-permeable BP-1-102 analog that targets STAT3 and STAT5 with comparable affinity.
包裝規格:10 MG
產品編號:4083613
純度規格:A depolymerized vanadate prepared from Sodium Orthovanadate with enhanced ability to competitively inhibit endogenous phosphatases.
包裝規格:5 ML,1 SET
產品編號:4083611
純度規格:A cell-permeable compound that targets human Replication Protein A (RPA) and inhibits its DNA-binding activity (IC50= 12.9 μM).
包裝規格:25 MG
產品編號:4083609
純度規格:A cell-permeable, selective inhibitor of RIP3-selective kinase with >1,000-fold selectivity over a vast majority of more than 300 other kinases.
包裝規格:10 MG
產品編號:4083606
純度規格:A cell-permeable pharmacological chaperone to increase neuronal retromer levels. Improves Vps35-Vps29-Vps26 retromer complex stability.
包裝規格:25 MG
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