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產品編號:4083791
純度規格:A synthetic amide of all-trans retinoic acid (RA) that displays reduced toxicity relative to RA while maintaining significant biological activity.
CAS NO:65646-68-6
包裝規格:5 MG
產品編號:4083790
純度規格:The Caspase-9 Substrate II, Colorimetric serves as the substrate for Caspase-9.
包裝規格:5 MG
產品編號:4083789
純度規格:Induces the reversion of transformed phenotypes of v-H-ras-transformed NIH 3T3 cells at low concentration (12.5 μM).
CAS NO:520-36-5
包裝規格:5 MG
產品編號:4083787
純度規格:for Northern and Southern blotting, solution
包裝規格:5 ML,5 X 5 ML
產品編號:4083786
純度規格:The VEGFR Tyrosine Kinase Inhibitor II, also referenced under CAS 269390-69-4, controls the biological activity of VEGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:269390-69-4
包裝規格:5 MG
產品編號:4083785
純度規格:A cell-permeable and reversible naphthoyl fused benzimidazole compound that acts as a highly selective, potent, ATP-competitive inhibitor of Ca2+/CaM-KK.
CAS NO:52029-86-4
包裝規格:5 MG
產品編號:4083784
純度規格:A cell-permeable p53 inhibitor that exhibits 10-fold higher potency and 50% longer half-life than Pifithrin-α.
CAS NO:60477-38-5
包裝規格:5 MG
產品編號:4083782
純度規格:The Necrosis Inhibitor, IM-54, also referenced under CAS 861891-50-1, selectively blocks oxidative stress-induced necrotic cell death. This small molecule/inhibitor is primarily used for Cancer applications.
CAS NO:861891-50-1
包裝規格:5 MG
產品編號:4083781
純度規格:The IL-2Rα Antagonist, also referenced under CAS 1217448-66-2, controls the biological activity of IL-2Rα.
CAS NO:1217448-66-2
包裝規格:5 MG
產品編號:4083780
純度規格:The Flt-3 Inhibitor, also referenced under CAS 301305-73-7, controls the biological activity of Flt-3. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:301305-73-7
包裝規格:5 MG
產品編號:4083779
純度規格:The DNA-PK Inhibitor II, also referenced under CAS 154447-35-5, controls the biological activity of DNA-PK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:154447-35-5
包裝規格:5 MG
產品編號:4083778
純度規格:A selective inhibitor of MMP-13 (IC50 = 10 μM).
CAS NO:1188890-36-9
包裝規格:5 MG
產品編號:4083777
純度規格:The CDC25 Phosphatase Inhibitor II, NSC 663284, also referenced under CAS 383907-43-5, controls the biological activity of CDC25 Phosphatase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:383907-43-5
包裝規格:5 MG
產品編號:4083776
純度規格:The CDC25 Phosphatase Inhibitor I, BN82002, also referenced under CAS 396073-89-5, controls the biological activity of CDC25 Phosphatase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:396073-89-5
包裝規格:5 MG
產品編號:4083775
純度規格:The ATM/ATR Kinase Inhibitor, also referenced under CAS 905973-89-9, controls the biological activity of ATM/ATR Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:905973-89-9
包裝規格:5 MG
產品編號:4083773
純度規格:(±)-Blebbistatin, CAS 674289-55-5, is a cell-permeable, selective, and reversible inhibitor of nonmuscle myosin II. Blocks cell blebbing and disrupts cell migration & cytoKinesis in vertebrate cells.
CAS NO:674289-55-5
包裝規格:5 MG
產品編號:4083772
純度規格:The Tubulin Polymerization Inhibitor II, also referenced under CAS 1151995-69-5, acts as an effective anti-microtubule agent. This small molecule/inhibitor is primarily used for Cell Structure applications.
CAS NO:1151995-69-5
包裝規格:5 MG
產品編號:4083771
純度規格:The PTP CD45 Inhibitor, also referenced under CAS 345630-40-2, controls the biological activity of PTP CD45. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:345630-40-2
包裝規格:5 MG
產品編號:4083770
純度規格:The MMP-2 Inhibitor III, also referenced under CAS 704888-90-4, controls the biological activity of MMP-2. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
CAS NO:704888-90-4
包裝規格:5 MG
產品編號:4083769
純度規格:The MK2a Inhibitor, also referenced under CAS 41179-33-3, controls the biological activity of MK2a. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:41179-33-3
包裝規格:5 MG
產品編號:4083768
純度規格:The JNK Inhibitor VIII, also referenced under CAS 894804-07-0, controls the biological activity of JNK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:894804-07-0
包裝規格:5 MG
產品編號:4083767
純度規格:The IP6K Inhibitor, also referenced under CAS 519178-28-0, controls the biological activity of IP6K.
CAS NO:519178-28-0
包裝規格:5 MG
產品編號:4083765
純度規格:The Cdk9 Inhibitor II, also referenced under CAS 140651-18-9, controls the biological activity of Cdk9. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:140651-18-9
包裝規格:5 MG
產品編號:4083764
純度規格:The Cdk4 Inhibitor III, also referenced under CAS 265312-55-8, controls the biological activity of Cdk4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:265312-55-8
包裝規格:5 MG
產品編號:4083763
純度規格:The Cdk4 Inhibitor II, NSC 625987, also referenced under CAS 141992-47-4, controls the biological activity of Cdk4. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:141992-47-4
包裝規格:5 MG
產品編號:4083762
純度規格:The Cdk2/9 Inhibitor, also referenced under CAS 507487-89-0, controls the biological activity of Cdk2/9. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:507487-89-0
包裝規格:5 MG
產品編號:4083761
純度規格:The Cathepsin L Inhibitor II controls the biological activity of Cathepsin L. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
包裝規格:5 MG
產品編號:4083760
純度規格:The Casein Kinase II Inhibitor III, TBCA, also referenced under CAS 934358-00-6, controls the biological activity of Casein Kinase II. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
CAS NO:934358-00-6
包裝規格:5 MG
產品編號:4083759
純度規格:A boronic acid-based arginine analog that acts as a slow-binding, competitive transition state inhibitor of arginases I and II (Ki = 310 nM for human recombinant type II arginase, pH 7.5).
包裝規格:5 MG
產品編號:4083752
純度規格:A cell-permeable, highly potent antagonist of TRPM8 (IC50 = 10.9 nM in icilin evoked Ca2+ currents in HEK293 cells)
包裝規格:10 MG
產品編號:4083751
純度規格:A cell-permeable, active-site directed, acyl-donor substrate competitive inhibitor of transglutaminase 2 (TG2, Ki = 11 μM).
包裝規格:5 MG
產品編號:4083750
純度規格:Inhibits TNFα/β-stimulated biological activity by modulating, but not abolishing, TNF-TNFR interaction via direct TNF affinity interaction (KD = 110 nM).
包裝規格:10 MG
產品編號:4083748
純度規格:A cell-permeable, selective, highly potent, non-nucleotide competitive inhibitor of telomerase activity (IC50 = 93 nM in HeLa cells nuclear extracts).
CAS NO:321674-73-1
包裝規格:10 MG
產品編號:4083747
純度規格:
包裝規格:5 MG
產品編號:4083745
純度規格:
包裝規格:10 MG
產品編號:4083744
純度規格:
CAS NO:1441190-66-4
包裝規格:500 μG
產品編號:4083743
純度規格:A cell-permeable, brain permeant, potent, reversible, ATP competitive inhibitor of Cdk4 and Cdk6 (IC50 = 11, 9, and 15 nM for Cdk4/D1, Cdk4/D3 and Cdk6/D2, respectively).
CAS NO:827022-32-2
包裝規格:5 MG
產品編號:4083741
純度規格:A cell permeable, selective, sphingosine competitive inhibitor of spingosine Kinase -2 (IC50 = 4.3 μM).
包裝規格:10 MG
產品編號:4083740
純度規格:A peptidyl toxin from venom of African tarantula, Hysterocrates gigas that acts as a high affinity, reversible blocker of Cav2.3 (α1E, R-type) channels (IC50 = 15-30 nM).
CAS NO:203460-30-4
包裝規格:10 μG
產品編號:4083738
純度規格:A cell-permeable inhibitor of SKP2-dependent p27Kip1 ubiquitination. Selectively induces the accumulation SCFSKP2 substrates in multiple myeloma RPMI 8226 cells.
包裝規格:10 MG
產品編號:4083737
純度規格:
包裝規格:10 MG
產品編號:4083736
純度規格:A highly potent agonist of GABAB receptor. Shown to be about 10-times more potent than baclofen.
CAS NO:127729-35-5
包裝規格:10 MG
產品編號:4083734
純度規格:
包裝規格:10 MG
產品編號:4083725
純度規格:A cell-permeable racemic mixture of Halofuginone that inhibits of prolyl-tRNA synthetase.
CAS NO:64924-67-0
包裝規格:10 MG
產品編號:4083724
純度規格:A cell-permeable, selective inhibitor of protein arginine methyltransferase 1 (PRMT1; IC50 = 9.5 μM).
包裝規格:10 MG
產品編號:4083722
純度規格:
包裝規格:10 MG
產品編號:4083721
純度規格:A cell-permeable inhibitor of Wnt secretion from L-cell Wnt1/2/3/3a/6/7a/9a transfectants (IC50 from 50 pM to 1.1 nM).
CAS NO:1243244-14-5
包裝規格:5 MG
產品編號:4083717
純度規格:A rhodanine-derived, reversible, photoactivated, TrpA1-selective channel activator.
包裝規格:10 MG
產品編號:4083714
純度規格:A cell-permeable, highly potent and selective inhibitor of phosphodiesterase 5 (PDEV; IC50 = 270 pM).
包裝規格:5 MG
產品編號:4083710
純度規格:A cell-permeable compound that selectively downregulates the expression of p21 (~10 μM), independent of p53.expression, at either transcription or post-transcriptional level.
包裝規格:10 MG
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